2
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12145 | N-Desethyl Sunitinib | SU-11662 | VEGFR , PDGFR , c-Kit |
N-Desethyl Sunitinib (SU-11662) is a sunitinib metabolite. | |||
T74127 | N-Desethyl Sunitinib hydrochloride | ||
N-Desethyl Sunitinib (SU-12662) (hydrochloride), a metabolite of sunitinib, is a robust ATP-competitive inhibitor of VEGFR, PDGFRβ, and KIT, demonstrating inhibition constants (K i values) of 2, 9, 17, 8, and 4 nM for VE... |